CN107759517A — 一种甲苯磺酸索拉非尼晶型ⅰ的制备方法
Assigned to Guangzhou Baiyunshan Pharmaceutical Holdings Co Ltd Baiyunshan Pharmaceutical General Factory · Expires 2018-03-06 · 8y expired
What this patent protects
一种甲苯磺酸索拉非尼晶型Ⅰ的制备方法,将晶型Ⅱ的甲苯磺酸索拉非尼溶解于二甲基亚砜中至溶解完全,加入醇类溶剂,析晶,分离,即得。本发明使用的有机溶剂均毒性较小、可工业化供应、廉价易得,本发明对环境友好,生产方法简单,得到的甲苯磺酸索拉非尼晶型Ⅰ晶形稳定。
USPTO Abstract
一种甲苯磺酸索拉非尼晶型Ⅰ的制备方法,将晶型Ⅱ的甲苯磺酸索拉非尼溶解于二甲基亚砜中至溶解完全,加入醇类溶剂,析晶,分离,即得。本发明使用的有机溶剂均毒性较小、可工业化供应、廉价易得,本发明对环境友好,生产方法简单,得到的甲苯磺酸索拉非尼晶型Ⅰ晶形稳定。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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