CN Patent
CN107721985A — 喹唑啉类酪氨酸激酶抑制剂的晶型
Assigned to Shandong Xuanzhu Pharma Co Ltd · Expires 2018-02-23 · 8y expired
What this patent protects
喹唑啉类酪氨酸激酶抑制剂的晶型。本发明属于医药领域,具体涉及一种Pan‑HER酪氨酸激酶抑制剂,即式(I)所示化合物(E)‑N‑(4‑((3‑氯‑4‑氟苯基)氨基)‑7‑甲氧基喹唑啉‑6‑基)‑4‑(2‑氮杂螺环[3.3]庚烷‑2‑基)‑2‑丁烯酰胺的晶型A、其制备方法、药物组合物,以及其在制备用于治疗和/或预防过度增生性疾病或慢性阻塞性肺病的药物中的应用。
USPTO Abstract
喹唑啉类酪氨酸激酶抑制剂的晶型。本发明属于医药领域,具体涉及一种Pan‑HER酪氨酸激酶抑制剂,即式(I)所示化合物(E)‑N‑(4‑((3‑氯‑4‑氟苯基)氨基)‑7‑甲氧基喹唑啉‑6‑基)‑4‑(2‑氮杂螺环[3.3]庚烷‑2‑基)‑2‑丁烯酰胺的晶型A、其制备方法、药物组合物,以及其在制备用于治疗和/或预防过度增生性疾病或慢性阻塞性肺病的药物中的应用。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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