CN Patent
CN107641123A — 一种依鲁替尼及其关键中间体的制备新方法
Assigned to NANJING YIHUA PHARMACEUTICAL CO Ltd · Expires 2018-01-30 · 8y expired
What this patent protects
本发明涉及一种依鲁替尼及其关键中间体的制备新方法,避免了现有合成工艺较为严苛的反应条件,以及价格昂贵的起始物料和试剂。采用一锅化法反应合成关键中间体,简化了较为繁琐的后处理操作,降低了成本。获得的中间体纯度在99%以上,收率较高,操作简单,适于工业化生产。
USPTO Abstract
本发明涉及一种依鲁替尼及其关键中间体的制备新方法,避免了现有合成工艺较为严苛的反应条件,以及价格昂贵的起始物料和试剂。采用一锅化法反应合成关键中间体,简化了较为繁琐的后处理操作,降低了成本。获得的中间体纯度在99%以上,收率较高,操作简单,适于工业化生产。
Drugs covered by this patent
- Imbruvica (ibrutinib) · AbbVie
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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