CN Patent

CN107200716B — 苯并噁嗪类化合物及其制备方法与应用

Assigned to Peking University · Expires 2020-04-17 · 6y expired

What this patent protects

本发明公开了一种苯并噁嗪类化合物,结构如式(I)所示,或其药学上可接受的盐,式(I)中各取代基的定义详见说明书。此外,本发明还公开了该化合物或其药学上可接受的盐的制备方法和应用。本发明的苯并噁嗪类化合物具有MEK抑制功能,并且对非磷酸化MEK具有抑制作用,同时,毒性低,可用作抗肿瘤和抗病毒药物。

USPTO Abstract

本发明公开了一种苯并噁嗪类化合物,结构如式(I)所示,或其药学上可接受的盐,式(I)中各取代基的定义详见说明书。此外,本发明还公开了该化合物或其药学上可接受的盐的制备方法和应用。本发明的苯并噁嗪类化合物具有MEK抑制功能,并且对非磷酸化MEK具有抑制作用,同时,毒性低,可用作抗肿瘤和抗病毒药物。

Drugs covered by this patent

Patent Metadata

Patent number
CN107200716B
Jurisdiction
CN
Classification
Expires
2020-04-17
Drug substance claim
No
Drug product claim
No
Assignee
Peking University
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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