CN Patent
CN107200716B — 苯并噁嗪类化合物及其制备方法与应用
Assigned to Peking University · Expires 2020-04-17 · 6y expired
What this patent protects
本发明公开了一种苯并噁嗪类化合物,结构如式(I)所示,或其药学上可接受的盐,式(I)中各取代基的定义详见说明书。此外,本发明还公开了该化合物或其药学上可接受的盐的制备方法和应用。本发明的苯并噁嗪类化合物具有MEK抑制功能,并且对非磷酸化MEK具有抑制作用,同时,毒性低,可用作抗肿瘤和抗病毒药物。
USPTO Abstract
本发明公开了一种苯并噁嗪类化合物,结构如式(I)所示,或其药学上可接受的盐,式(I)中各取代基的定义详见说明书。此外,本发明还公开了该化合物或其药学上可接受的盐的制备方法和应用。本发明的苯并噁嗪类化合物具有MEK抑制功能,并且对非磷酸化MEK具有抑制作用,同时,毒性低,可用作抗肿瘤和抗病毒药物。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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