CN Patent
CN107056706B — 一种用于制备盐酸伊伐布雷定α晶型的方法
Assigned to Shanghai Maijin Biomedical Technology Co ltd · Expires 2020-05-05 · 6y expired
What this patent protects
本发明涉及一种用于制备盐酸伊伐布雷定α晶型的方法。具体而言,本发明涉及式I所示的盐酸伊伐布雷定α晶型的制备方法,其特征是盐酸伊伐布雷定的无定形或其他晶型在甲苯、乙酸丁酯或4‑甲基‑2‑戊酮等高沸点不良溶剂中高温搅拌转晶。利用本法制备盐酸伊伐布雷定α晶型,操作过程简便,产品收率高、易干燥。
USPTO Abstract
本发明涉及一种用于制备盐酸伊伐布雷定α晶型的方法。具体而言,本发明涉及式I所示的盐酸伊伐布雷定α晶型的制备方法,其特征是盐酸伊伐布雷定的无定形或其他晶型在甲苯、乙酸丁酯或4‑甲基‑2‑戊酮等高沸点不良溶剂中高温搅拌转晶。利用本法制备盐酸伊伐布雷定α晶型,操作过程简便,产品收率高、易干燥。
Drugs covered by this patent
- Corlanor (IVABRADINE) · Amgen
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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