CN106994119A — 含有依匹哌唑或其盐的口腔崩解片及其制备方法
Assigned to Zhejiang Huahai Pharmaceutical Co Ltd · Expires 2017-08-01 · 9y expired
What this patent protects
本发明涉及一种含有依匹哌唑或其盐的口腔崩解片,还涉及其制备方法。该口腔崩解片含有:0.06%~15.0%的依匹哌唑;40.0%~95.0%的赋形剂;3.0%~50.0%的崩解剂;0.0%~6.0%的润滑剂;0.05%~5.0%的矫味剂。该口腔崩解片是通过先将活性成分依匹哌唑制备成固体分散体,然后与其它辅料混合制备得到的。所述口腔崩解片具备崩解迅速,口感好,生物利用度高,质量稳定可控,辅料安全易得,制备方法简单,无需昂贵特殊设备,易贮藏,易运输的优点。
USPTO Abstract
本发明涉及一种含有依匹哌唑或其盐的口腔崩解片,还涉及其制备方法。该口腔崩解片含有:0.06%~15.0%的依匹哌唑;40.0%~95.0%的赋形剂;3.0%~50.0%的崩解剂;0.0%~6.0%的润滑剂;0.05%~5.0%的矫味剂。该口腔崩解片是通过先将活性成分依匹哌唑制备成固体分散体,然后与其它辅料混合制备得到的。所述口腔崩解片具备崩解迅速,口感好,生物利用度高,质量稳定可控,辅料安全易得,制备方法简单,无需昂贵特殊设备,易贮藏,易运输的优点。
Drugs covered by this patent
- Rexulti (BREXPIPRAZOLE) · Otsuka
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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