CN Patent
CN106905294A — 5‑[2,6‑二(4‑吗啉基)‑4‑嘧啶基]‑4‑(三氟甲基)‑2‑吡啶胺的晶型及其制备方法
Assigned to Suzhou Best Pharmaceutical Co Ltd · Expires 2017-06-30 · 9y expired
What this patent protects
本发明涉及5‑[2,6‑二(4‑吗啉基)‑4‑嘧啶基]‑4‑(三氟甲基)‑2‑吡啶胺的晶型及其制备方法,具体地为晶型A和晶型C。本发明提供的晶型稳定性良好、溶解度更高、引湿性较低,对未来该药物的优化和开发具有重要价值。
USPTO Abstract
本发明涉及5‑[2,6‑二(4‑吗啉基)‑4‑嘧啶基]‑4‑(三氟甲基)‑2‑吡啶胺的晶型及其制备方法,具体地为晶型A和晶型C。本发明提供的晶型稳定性良好、溶解度更高、引湿性较低,对未来该药物的优化和开发具有重要价值。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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