CN Patent
CN106883212A — 一种xli晶型阿昔替尼的制备方法
Assigned to HEFEI TOPWAY BIOTECHNOLOGY CO Ltd · Expires 2017-06-23 · 9y expired
What this patent protects
本发明公开了一种XLI晶型阿昔替尼的制备方法,其特征在于,包括如下步骤:S1、在避光环境中,将阿昔替尼、质子性溶剂混匀,重结晶,干燥得到中间体;S2、在避光环境中,取S1得到的中间体在无水溶剂中进行加晶种重结晶得到XLI晶型阿昔替尼。本发明操作简便,重复性高,成本低,收率高,适合工业化生产。
USPTO Abstract
本发明公开了一种XLI晶型阿昔替尼的制备方法,其特征在于,包括如下步骤:S1、在避光环境中,将阿昔替尼、质子性溶剂混匀,重结晶,干燥得到中间体;S2、在避光环境中,取S1得到的中间体在无水溶剂中进行加晶种重结晶得到XLI晶型阿昔替尼。本发明操作简便,重复性高,成本低,收率高,适合工业化生产。
Drugs covered by this patent
- Inlyta (Axitinib) · Pfizer
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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