CN Patent
CN106866624B — 一种卡比替尼的化学合成方法
Assigned to JINING MEDICAL COLLEGE · Expires 2017-12-26 · 8y expired
What this patent protects
本发明属于化学合成领域,具体涉及一种卡比替尼的制备方法。该方法以2,3,4‑三氟苯甲酸苄酯为起始原料,通过取代反应、脱保护反应、酰胺化反应、催化加成反应等步骤得到卡比替尼。该方法原料价廉易得,工艺路线段,工反应过程易于操作,收率高,且环境友好,适合工业化大批量生产。
USPTO Abstract
本发明属于化学合成领域,具体涉及一种卡比替尼的制备方法。该方法以2,3,4‑三氟苯甲酸苄酯为起始原料,通过取代反应、脱保护反应、酰胺化反应、催化加成反应等步骤得到卡比替尼。该方法原料价廉易得,工艺路线段,工反应过程易于操作,收率高,且环境友好,适合工业化大批量生产。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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