CN106794185A — Rucaparib的高剂量强度片剂
Assigned to Clovis Oncology Inc · Expires 2017-05-31 · 9y expired
What this patent protects
本发明公开包含高剂量的8‑氟‑2‑{4‑[(甲基氨基)甲基]苯基}‑1,3,4,5‑四氢‑6H‑氮杂 并[5,4,3‑cd]吲哚‑6‑酮樟脑磺酸盐的片剂。本发明涉及rucaparib的高剂量强度片剂。在一些实施方案中,所述片剂包含45‑90%w/w的rucaparib樟脑磺酸盐。在一些实施方案中,所述干法制粒片剂包含45‑90%w/w的rucaparib樟脑磺酸盐。一个这样的实施方案是包含至少200mg rucaparib的片剂。另一实施方案是包含至少300mg rucaparib的片剂。
USPTO Abstract
本发明公开包含高剂量的8‑氟‑2‑{4‑[(甲基氨基)甲基]苯基}‑1,3,4,5‑四氢‑6H‑氮杂 并[5,4,3‑cd]吲哚‑6‑酮樟脑磺酸盐的片剂。本发明涉及rucaparib的高剂量强度片剂。在一些实施方案中,所述片剂包含45‑90%w/w的rucaparib樟脑磺酸盐。在一些实施方案中,所述干法制粒片剂包含45‑90%w/w的rucaparib樟脑磺酸盐。一个这样的实施方案是包含至少200mg rucaparib的片剂。另一实施方案是包含至少300mg rucaparib的片剂。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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