CN Patent
CN106432209A — Lumacaftor的新晶型及其制备方法
Assigned to Crystal Pharmatech Co Ltd · Expires 2017-02-22 · 9y expired
What this patent protects
本发明提供lumacaftor的晶型A及其制备方法。本发明提供的晶型A的X射线粉末衍射图在2theta值为8.8°±0.2°、21.2°±0.2°、22.2°±0.2°处具有特征峰。本发明的晶型A稳定性好,比之现有技术溶解度更高,对未来该药物的优化和开发具有重要价值。
USPTO Abstract
本发明提供lumacaftor的晶型A及其制备方法。本发明提供的晶型A的X射线粉末衍射图在2theta值为8.8°±0.2°、21.2°±0.2°、22.2°±0.2°处具有特征峰。本发明的晶型A稳定性好,比之现有技术溶解度更高,对未来该药物的优化和开发具有重要价值。
Drugs covered by this patent
- Kalydeco (IVACAFTOR) · Vertex Pharms Inc
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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