CN Patent
CN106432197B — 一种雷迪帕韦中间体单对甲苯磺酸盐、其晶型及其制备方法
Assigned to SHANGHAI FOREFRONT PHARMA · Expires 2019-12-10 · 6y expired
What this patent protects
本发明公开了一种雷迪帕韦中间体单对甲苯磺酸盐、其晶型及其制备方法。本发明所提供的制备方法制得的晶型A具有良好的化学纯度和产品质量,制备方法简单、快速,便于大规模化生产。同时,晶型A具有非常高的纯度,特别适合用作生产雷迪帕韦的中间体,从而提高终产物雷迪帕韦的质量,并减少杂质。
USPTO Abstract
本发明公开了一种雷迪帕韦中间体单对甲苯磺酸盐、其晶型及其制备方法。本发明所提供的制备方法制得的晶型A具有良好的化学纯度和产品质量,制备方法简单、快速,便于大规模化生产。同时,晶型A具有非常高的纯度,特别适合用作生产雷迪帕韦的中间体,从而提高终产物雷迪帕韦的质量,并减少杂质。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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