CN Patent
CN106336403A — 依帕列净的工业制备方法
Assigned to Jiangsu Hansoh Pharmaceutical Group Co Ltd · Expires 2017-01-18 · 9y expired
What this patent protects
本发明公开了依帕列净的工业制备方法。具体地,本发明涉及下式所示依帕列净即(1S)‑1,5‑脱水‑1‑(4‑氯‑3‑{4‑[(3S)‑四氢呋喃‑3‑基氧基]苄基}苯基)‑D‑葡萄糖醇的制备方法,且包含在该方法中所获得的中间体。本发明所提供的依帕列净生产工艺稳定,可重现性好,适合规模化生产。
USPTO Abstract
本发明公开了依帕列净的工业制备方法。具体地,本发明涉及下式所示依帕列净即(1S)‑1,5‑脱水‑1‑(4‑氯‑3‑{4‑[(3S)‑四氢呋喃‑3‑基氧基]苄基}苯基)‑D‑葡萄糖醇的制备方法,且包含在该方法中所获得的中间体。本发明所提供的依帕列净生产工艺稳定,可重现性好,适合规模化生产。
Drugs covered by this patent
- Jardiance (empagliflozin) · Boehringer Ingelheim
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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