CN Patent

CN106279134A — 卡格列净单晶及其制备方法和用途

Assigned to Waterstone Pharmaceuticals Wuhan Co Ltd · Expires 2017-01-04 · 9y expired

What this patent protects

本发明涉及一种卡格列净单晶及其制备方法和用途,述卡格列净单晶的X射线粉末衍射在衍射角2θ=7.95,10.92,13.94,15.46,15.94,18.82,20.27,22.72和26.78度处有特征峰,所得单晶未见报道,测定其晶体结构属斜方晶系,空间群为P2(1)2(1)2(1),晶包内分子数Z=4,常温下为无色针状结晶,形态良好,纯度高达99%;其制备方法使得卡格列净与其他杂质实现良好的分离,且重现性好。

USPTO Abstract

本发明涉及一种卡格列净单晶及其制备方法和用途,述卡格列净单晶的X射线粉末衍射在衍射角2θ=7.95,10.92,13.94,15.46,15.94,18.82,20.27,22.72和26.78度处有特征峰,所得单晶未见报道,测定其晶体结构属斜方晶系,空间群为P2(1)2(1)2(1),晶包内分子数Z=4,常温下为无色针状结晶,形态良好,纯度高达99%;其制备方法使得卡格列净与其他杂质实现良好的分离,且重现性好。

Drugs covered by this patent

Patent Metadata

Patent number
CN106279134A
Jurisdiction
CN
Classification
Expires
2017-01-04
Drug substance claim
No
Drug product claim
No
Assignee
Waterstone Pharmaceuticals Wuhan Co Ltd
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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