CN106031710B — 一种富马酸氟呐普拉赞的注射剂及其制备方法
Assigned to Nanjing Yoko Biological Pharmaceutical Group Co Ltd · Expires 2019-03-12 · 7y expired
What this patent protects
本发明属于药物制剂技术领域,尤其涉及一种具有治疗胃酸相关性疾病作用的钾离子竞争性酸阻滞剂:富马酸氟呐普拉赞的注射剂及其制备方法。本发明克服了主药富马酸氟呐普拉赞的水溶性差的缺陷,采用磺丁基醚‑β‑环糊精或者羟丙基‑β‑环糊精的包合形式进行増溶,制备所得的注射剂具有稳定性好,安全性高,长期放置不沉淀等优势,能够满足不方便口服给药病人的用药需求。
USPTO Abstract
本发明属于药物制剂技术领域,尤其涉及一种具有治疗胃酸相关性疾病作用的钾离子竞争性酸阻滞剂:富马酸氟呐普拉赞的注射剂及其制备方法。本发明克服了主药富马酸氟呐普拉赞的水溶性差的缺陷,采用磺丁基醚‑β‑环糊精或者羟丙基‑β‑环糊精的包合形式进行増溶,制备所得的注射剂具有稳定性好,安全性高,长期放置不沉淀等优势,能够满足不方便口服给药病人的用药需求。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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