CN Patent
CN105777651A — 聚腺苷酸二磷酸核糖转移酶抑制剂的晶型及其制备方法和医药用途
Assigned to Jiangsu Hansoh Pharmaceutical Group Co Ltd · Expires 2016-07-20 · 10y expired
What this patent protects
本发明涉及聚腺苷酸二磷酸核糖转移酶抑制剂的晶型及其制备方法和医药用途。具体涉及聚腺苷酸二磷酸核糖转移酶(PARP)抑制剂即4‐[3‐(4‐环丙烷羰基‐哌嗪‐1‐羰基)‐4‐氟‐苄基]‐2H‐酞嗪‐1‐酮的一种新晶型、其制备方法、药物组合物和在治疗癌症中的用途,本发明所提供的新晶型重现性好,稳定易得,适合药物开发。
USPTO Abstract
本发明涉及聚腺苷酸二磷酸核糖转移酶抑制剂的晶型及其制备方法和医药用途。具体涉及聚腺苷酸二磷酸核糖转移酶(PARP)抑制剂即4‐[3‐(4‐环丙烷羰基‐哌嗪‐1‐羰基)‐4‐氟‐苄基]‐2H‐酞嗪‐1‐酮的一种新晶型、其制备方法、药物组合物和在治疗癌症中的用途,本发明所提供的新晶型重现性好,稳定易得,适合药物开发。
Drugs covered by this patent
- Lynparza (olaparib) · AstraZeneca
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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