CN Patent
CN105753944B — 达卡他韦及其衍生物的制备中间体
Assigned to Chia Tai Tianqing Pharmaceutical Group Co Ltd · Expires 2019-10-01 · 7y expired
What this patent protects
本发明属于药物化学领域,具体涉及达卡他韦及其衍生物的制备中间体,以及它们的制备方法。该制备方法不仅简化了后处理过程,还出乎意料地提高每步反应的收率,进而提高了路线的总收率。此外,还提高了原料的利用率,节约成本,更适应工业化大生产。
USPTO Abstract
本发明属于药物化学领域,具体涉及达卡他韦及其衍生物的制备中间体,以及它们的制备方法。该制备方法不仅简化了后处理过程,还出乎意料地提高每步反应的收率,进而提高了路线的总收率。此外,还提高了原料的利用率,节约成本,更适应工业化大生产。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
Track this patent
Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.