CN Patent

CN105753944B — 达卡他韦及其衍生物的制备中间体

Assigned to Chia Tai Tianqing Pharmaceutical Group Co Ltd · Expires 2019-10-01 · 7y expired

What this patent protects

本发明属于药物化学领域,具体涉及达卡他韦及其衍生物的制备中间体,以及它们的制备方法。该制备方法不仅简化了后处理过程,还出乎意料地提高每步反应的收率,进而提高了路线的总收率。此外,还提高了原料的利用率,节约成本,更适应工业化大生产。

USPTO Abstract

本发明属于药物化学领域,具体涉及达卡他韦及其衍生物的制备中间体,以及它们的制备方法。该制备方法不仅简化了后处理过程,还出乎意料地提高每步反应的收率,进而提高了路线的总收率。此外,还提高了原料的利用率,节约成本,更适应工业化大生产。

Drugs covered by this patent

Patent Metadata

Patent number
CN105753944B
Jurisdiction
CN
Classification
Expires
2019-10-01
Drug substance claim
No
Drug product claim
No
Assignee
Chia Tai Tianqing Pharmaceutical Group Co Ltd
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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