CN Patent

CN105753867B — 一种改进的阿维巴坦钠中间体化合物的制备方法

Assigned to QILU PHARMACEUTICAL (HAINAN) CO Ltd · Expires 2018-03-27 · 8y expired

What this patent protects

本发明属于医药化学技术领域,具体涉及一种β‑内酰胺酶抑制剂药物阿维巴坦钠及其中间体的制备方法。本发明采用三乙基硅烷实现苄基脱除,免了现有技术中的氢化催化操作,使得反应条件更加温和,降低了安全风险,大大提高了产品收率和纯度,更适合规模化生产。

USPTO Abstract

本发明属于医药化学技术领域,具体涉及一种β‑内酰胺酶抑制剂药物阿维巴坦钠及其中间体的制备方法。本发明采用三乙基硅烷实现苄基脱除,免了现有技术中的氢化催化操作,使得反应条件更加温和,降低了安全风险,大大提高了产品收率和纯度,更适合规模化生产。

Drugs covered by this patent

Patent Metadata

Patent number
CN105753867B
Jurisdiction
CN
Classification
Expires
2018-03-27
Drug substance claim
No
Drug product claim
No
Assignee
QILU PHARMACEUTICAL (HAINAN) CO Ltd
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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