CN Patent
CN105646484A — 晶型b及制备方法
Assigned to Individual · Expires 2016-06-08 · 10y expired
What this patent protects
本发明公开晶型B,其特征在于,使用Cu-Kα辐射,以2θ角度表示的X-射线粉末衍射(X-RPD)在6.4±0.2°,7.9±0.2°,8.7±0.2°,9.8±0.2°,10.0±0.2°,17.0±0.2°处有衍射峰。本发明所述的晶型B可安全地大规模制备并纯化,且储存稳定,不具有吸湿性,非常适用于制备吸入性制剂,与乳糖和淀粉等赋形剂的兼容性好。
USPTO Abstract
本发明公开晶型B,其特征在于,使用Cu-Kα辐射,以2θ角度表示的X-射线粉末衍射(X-RPD)在6.4±0.2°,7.9±0.2°,8.7±0.2°,9.8±0.2°,10.0±0.2°,17.0±0.2°处有衍射峰。本发明所述的晶型B可安全地大规模制备并纯化,且储存稳定,不具有吸湿性,非常适用于制备吸入性制剂,与乳糖和淀粉等赋形剂的兼容性好。
Drugs covered by this patent
- Imbruvica (ibrutinib) · AbbVie
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
Track this patent
Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.