CN Patent
CN105616418A — 含有细胞周期蛋白抑制剂的药物制剂及其制备方法
Assigned to Jiangsu Hansoh Pharmaceutical Group Co Ltd · Expires 2016-06-01 · 10y expired
What this patent protects
本发明公开了含有细胞周期蛋白抑制剂的药物制剂及其制备方法。具体地,本发明涉及一种以式Ⅰ所示的6-乙酰基-8-环戊基-5-甲基-2-(5-哌嗪-1-基-吡啶-2-基氨基)-8H-吡啶并[2,3-d]嘧啶-7-酮或其盐为活性成分的药物制剂,所述盐包括盐酸盐、羟乙基磺酸盐,所述药物剂型包括片剂、胶囊剂。所述剂型均具有良好的稳定性以及优异的溶出行为。
USPTO Abstract
本发明公开了含有细胞周期蛋白抑制剂的药物制剂及其制备方法。具体地,本发明涉及一种以式Ⅰ所示的6-乙酰基-8-环戊基-5-甲基-2-(5-哌嗪-1-基-吡啶-2-基氨基)-8H-吡啶并[2,3-d]嘧啶-7-酮或其盐为活性成分的药物制剂,所述盐包括盐酸盐、羟乙基磺酸盐,所述药物剂型包括片剂、胶囊剂。所述剂型均具有良好的稳定性以及优异的溶出行为。
Drugs covered by this patent
- Palbociclib (palbociclib) · Pfizer Inc.
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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