CN Patent
CN105481757A — 一种哌马色林的制备方法
Assigned to BEIJING KANG LISHENG PHARMACEUTICAL TECHNOLOGY DEVELOPMENT Co Ltd · Expires 2016-04-13 · 10y expired
What this patent protects
本发明涉及一种哌马色林的制备方法,以4-氟苄胺为起始原料,先与N-甲基-4-哌啶酮还原胺化,再与氯甲酸苄酯进行对接,最后与4-异丁氧基苄胺反应,制备得到哌马色林。此制备方法简便易行、收率高,质量好,便于工业化生产。
USPTO Abstract
本发明涉及一种哌马色林的制备方法,以4-氟苄胺为起始原料,先与N-甲基-4-哌啶酮还原胺化,再与氯甲酸苄酯进行对接,最后与4-异丁氧基苄胺反应,制备得到哌马色林。此制备方法简便易行、收率高,质量好,便于工业化生产。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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