CN Patent

CN105457038A — 一种速释型药物磷脂化合物及其药物组合物

Assigned to Southeast University · Expires 2016-04-06 · 10y expired

What this patent protects

本发明公开了一种速释型药物磷脂化合物及其药物组合物,该化合物中,药物Y 1 、Y 2 通过化学键与速释型疏水间隔臂和增强型疏水间隔臂相连,两种间隔臂相互协同增强疏水作用,构成疏水亲脂链;两条疏水链与磷脂亲水头相连,构成两亲性分子。药物组合物为速释型药物磷脂化合物或该化合物和药效学上可接受的载体的组合药物组合物。该速释型药物磷脂化合物及其脂质体纳米颗粒可用作液体制剂、固体制剂、半固体制剂、灭菌制剂和无菌制剂,毒性低,可用于各种肿瘤等疾病的高效治疗。

USPTO Abstract

本发明公开了一种速释型药物磷脂化合物及其药物组合物,该化合物中,药物Y 1 、Y 2 通过化学键与速释型疏水间隔臂和增强型疏水间隔臂相连,两种间隔臂相互协同增强疏水作用,构成疏水亲脂链;两条疏水链与磷脂亲水头相连,构成两亲性分子。药物组合物为速释型药物磷脂化合物或该化合物和药效学上可接受的载体的组合药物组合物。该速释型药物磷脂化合物及其脂质体纳米颗粒可用作液体制剂、固体制剂、半固体制剂、灭菌制剂和无菌制剂,毒性低,可用于各种肿瘤等疾病的高效治疗。

Drugs covered by this patent

Patent Metadata

Patent number
CN105457038A
Jurisdiction
CN
Classification
Expires
2016-04-06
Drug substance claim
No
Drug product claim
No
Assignee
Southeast University
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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