CN Patent
CN105348265A — 一种具有ALK和c-Met抑制活性的2,4-二取代杂环三氮唑类化合物的制备和应用
Assigned to Individual · Expires 2016-02-24 · 10y expired
What this patent protects
本发明涉及式(I)2,4-二取代杂环三氮唑类化合物的制备及其应用,其中R1和R2的定义见说明书。本发明提供的式(I)化合物是ALK和c-Met激酶抑制剂,通过阻断信号通路,终止下游信号级联通路,发挥抑制癌细胞增殖的作用。式(I)化合物可作为潜在的抗癌治疗药物。
USPTO Abstract
本发明涉及式(I)2,4-二取代杂环三氮唑类化合物的制备及其应用,其中R1和R2的定义见说明书。本发明提供的式(I)化合物是ALK和c-Met激酶抑制剂,通过阻断信号通路,终止下游信号级联通路,发挥抑制癌细胞增殖的作用。式(I)化合物可作为潜在的抗癌治疗药物。
Drugs covered by this patent
- Xalkori (crizotinib) · Pfizer
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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