CN Patent
CN105315263B — 阿法替尼中间体的合成方法
Assigned to Chia Tai Tianqing Pharmaceutical Group Co Ltd · Expires 2018-11-27 · 7y expired
What this patent protects
本发明涉及阿法替尼中间体的合成方法,该方法由(S)‑N‑(3‑氯‑4‑氟苯基)‑6‑硝基‑7‑[(四氢呋喃‑3‑基)氧基]喹唑啉‑4‑胺与保险粉反应得到,本发明的方法不仅获得高的产率,而且简化反应的后处理。
USPTO Abstract
本发明涉及阿法替尼中间体的合成方法,该方法由(S)‑N‑(3‑氯‑4‑氟苯基)‑6‑硝基‑7‑[(四氢呋喃‑3‑基)氧基]喹唑啉‑4‑胺与保险粉反应得到,本发明的方法不仅获得高的产率,而且简化反应的后处理。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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