CN Patent
CN105111215B — 一种周期蛋白依赖性激酶抑制剂的晶型及其制备方法
Assigned to SUZHOU PENGXU PHARMATECH Co Ltd · Expires 2019-06-18 · 7y expired
What this patent protects
本发明涉及7‑环戊基‑2‑(5‑哌嗪‑1‑基‑吡啶‑2‑基氨基)‑7H‑吡咯并[2,3‑D]嘧啶‑6‑羧酸二甲酰胺的的半琥珀酸盐的新晶型及其制备方法,单琥珀酸盐的新晶型及其制备方法。本发明的式(I)化合物的半琥珀酸盐新晶型,单琥珀酸盐新晶型,具有良好的稳定性、较低的引湿性、工艺可开发和易处理性等有利性能,且制备方法简单,成本低廉,对未来该药物的优化和开发具有重要价值。
USPTO Abstract
本发明涉及7‑环戊基‑2‑(5‑哌嗪‑1‑基‑吡啶‑2‑基氨基)‑7H‑吡咯并[2,3‑D]嘧啶‑6‑羧酸二甲酰胺的的半琥珀酸盐的新晶型及其制备方法,单琥珀酸盐的新晶型及其制备方法。本发明的式(I)化合物的半琥珀酸盐新晶型,单琥珀酸盐新晶型,具有良好的稳定性、较低的引湿性、工艺可开发和易处理性等有利性能,且制备方法简单,成本低廉,对未来该药物的优化和开发具有重要价值。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
Track this patent
Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.