CN Patent
CN105061506B — 抗肿瘤药物ap26113的制备方法
Assigned to Shaoxing baiweikang Biotechnology Co.,Ltd. · Expires 2017-08-29 · 9y expired
What this patent protects
本发明揭示了一种抗肿瘤药物AP26113(I)的制备方法,其制备步骤包括:N‑[2‑甲氧基‑4‑[4‑(二甲基氨基)哌啶‑1‑基]苯胺]胍依次与N,N‑二甲氨基丙烯酸酯、4‑(二甲基亚磷酰)苯胺和氯化剂发生环合反应、缩合反应以及氯化反应制得AP26113(I)。该制备方法原料易得,副反应少,经济环保,适合工业化生产。
USPTO Abstract
本发明揭示了一种抗肿瘤药物AP26113(I)的制备方法,其制备步骤包括:N‑[2‑甲氧基‑4‑[4‑(二甲基氨基)哌啶‑1‑基]苯胺]胍依次与N,N‑二甲氨基丙烯酸酯、4‑(二甲基亚磷酰)苯胺和氯化剂发生环合反应、缩合反应以及氯化反应制得AP26113(I)。该制备方法原料易得,副反应少,经济环保,适合工业化生产。
Drugs covered by this patent
- Alunbrig (brigatinib) · Takeda
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
Track this patent
Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.