CN Patent

CN105061506B — 抗肿瘤药物ap26113的制备方法

Assigned to Shaoxing baiweikang Biotechnology Co.,Ltd. · Expires 2017-08-29 · 9y expired

What this patent protects

本发明揭示了一种抗肿瘤药物AP26113(I)的制备方法,其制备步骤包括:N‑[2‑甲氧基‑4‑[4‑(二甲基氨基)哌啶‑1‑基]苯胺]胍依次与N,N‑二甲氨基丙烯酸酯、4‑(二甲基亚磷酰)苯胺和氯化剂发生环合反应、缩合反应以及氯化反应制得AP26113(I)。该制备方法原料易得,副反应少,经济环保,适合工业化生产。

USPTO Abstract

本发明揭示了一种抗肿瘤药物AP26113(I)的制备方法,其制备步骤包括:N‑[2‑甲氧基‑4‑[4‑(二甲基氨基)哌啶‑1‑基]苯胺]胍依次与N,N‑二甲氨基丙烯酸酯、4‑(二甲基亚磷酰)苯胺和氯化剂发生环合反应、缩合反应以及氯化反应制得AP26113(I)。该制备方法原料易得,副反应少,经济环保,适合工业化生产。

Drugs covered by this patent

Patent Metadata

Patent number
CN105061506B
Jurisdiction
CN
Classification
Expires
2017-08-29
Drug substance claim
No
Drug product claim
No
Assignee
Shaoxing baiweikang Biotechnology Co.,Ltd.
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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