CN Patent
CN105030685B — 一种恩杂鲁胺固体分散体口服制剂
Assigned to FERGUSON (WUHAN) BIOTECHNOLOGY Co Ltd · Expires 2018-02-27 · 8y expired
What this patent protects
本发明公开了一种恩杂鲁胺固体分散体的口服制剂,含有有效剂量的恩杂鲁胺,还含有用于分散恩杂鲁胺的水溶性聚合物载体,所述恩杂鲁胺与水溶性聚合物载体的质量比为1∶0.5~3。本发明有效地提高了制剂中恩杂鲁胺的溶解度和溶出度,从而提高了恩杂鲁胺的生物利用度,同时还提高了恩杂鲁胺的质量稳定性和安全性。
USPTO Abstract
本发明公开了一种恩杂鲁胺固体分散体的口服制剂,含有有效剂量的恩杂鲁胺,还含有用于分散恩杂鲁胺的水溶性聚合物载体,所述恩杂鲁胺与水溶性聚合物载体的质量比为1∶0.5~3。本发明有效地提高了制剂中恩杂鲁胺的溶解度和溶出度,从而提高了恩杂鲁胺的生物利用度,同时还提高了恩杂鲁胺的质量稳定性和安全性。
Drugs covered by this patent
- Xtandi (enzalutamide) · Astellas Pharma
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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