CN Patent
CN104926669A — 反式-4-二甲基胺基巴豆酸盐酸盐的制备方法
Assigned to Jiangsu Hansoh Pharmaceutical Group Co Ltd · Expires 2015-09-23 · 11y expired
What this patent protects
本发明涉及反式-4-二甲基胺基巴豆酸盐酸盐的制备方法,其是一种重要医药中间体式(I)的制备过程,4-溴代巴豆酸甲酯和二甲胺类化合物经过取代、成盐、水解、成盐制得式(I)化合物反式-4-二甲基胺基巴豆酸盐酸盐。该制备方法工艺简洁、收率高,适合工业化放大的要求。
USPTO Abstract
本发明涉及反式-4-二甲基胺基巴豆酸盐酸盐的制备方法,其是一种重要医药中间体式(I)的制备过程,4-溴代巴豆酸甲酯和二甲胺类化合物经过取代、成盐、水解、成盐制得式(I)化合物反式-4-二甲基胺基巴豆酸盐酸盐。该制备方法工艺简洁、收率高,适合工业化放大的要求。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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