CN Patent
CN104840965B — 波生坦的制剂及其稳定剂
Assigned to Chongqing Huapont Pharm Co Ltd · Expires 2018-05-08 · 8y expired
What this patent protects
本发明属于药物制剂领域,特别涉及波生坦药物制剂的组合物,该组合物包含波生坦、一水乳糖、微晶纤维素KG802,十二烷基硫酸钠或吐温‑80。所述组合物增加了波生坦的溶出度,提高了制剂晶型稳定性。该组合物可制备成片剂、胶囊剂、颗粒剂等固体口服制剂,制备方法简单、可行、易于实现产业化大生产。
USPTO Abstract
本发明属于药物制剂领域,特别涉及波生坦药物制剂的组合物,该组合物包含波生坦、一水乳糖、微晶纤维素KG802,十二烷基硫酸钠或吐温‑80。所述组合物增加了波生坦的溶出度,提高了制剂晶型稳定性。该组合物可制备成片剂、胶囊剂、颗粒剂等固体口服制剂,制备方法简单、可行、易于实现产业化大生产。
Drugs covered by this patent
- Tracleer (BOSENTAN) · AstraZeneca
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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