CN Patent

CN104736178A — 布鲁顿酪氨酸激酶抑制剂的晶形

Assigned to Pharmacyclics LLC · Expires 2015-06-24 · 11y expired

What this patent protects

本文描述了布鲁顿酪氨酸激酶(Btk)抑制剂1-((R)-3-(4-氨基-3-(4-苯氧基苯基)-1H-吡唑并[3,4-d]嘧啶-1-基)哌啶-1-基)丙-2-烯-1-酮,包括其晶形、溶剂化物和药学上可接的盐。还公开了包含该Btk抑制剂的药物组合物,以及单独地或与其他治疗剂联合地使用该Btk抑制剂治疗自身免疫疾病或状况、异种免疫疾病或状况、包括淋巴瘤在内的癌症以及炎性疾病或状况的方法。

USPTO Abstract

本文描述了布鲁顿酪氨酸激酶(Btk)抑制剂1-((R)-3-(4-氨基-3-(4-苯氧基苯基)-1H-吡唑并[3,4-d]嘧啶-1-基)哌啶-1-基)丙-2-烯-1-酮,包括其晶形、溶剂化物和药学上可接的盐。还公开了包含该Btk抑制剂的药物组合物,以及单独地或与其他治疗剂联合地使用该Btk抑制剂治疗自身免疫疾病或状况、异种免疫疾病或状况、包括淋巴瘤在内的癌症以及炎性疾病或状况的方法。

Drugs covered by this patent

Patent Metadata

Patent number
CN104736178A
Jurisdiction
CN
Classification
Expires
2015-06-24
Drug substance claim
No
Drug product claim
No
Assignee
Pharmacyclics LLC
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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