CN Patent
CN104710345B — 用于制备4‑(2‑(4‑甲基苯基硫基))苯基哌啶的化合物、其制备方法及应用
Assigned to Nhwa Pharmaceutical Corp · Expires 2017-09-05 · 9y expired
What this patent protects
本发明公开了用于制备4‑(2‐(4‐甲基苯基硫基))苯基哌啶的化合物、其制备方法及应用。本发明提供了两种制备4‑(2‐(4‐甲基苯基巯基))苯基哌啶的中间体:3‑(2‐(4‐甲基苯基巯基))苯基戊二酸和4‑(2‐(4‐甲基苯基巯基))苯基哌啶‐2,6‐二酮及其制备与应用。该方法收率高,操作安全、方便,对环境污染小且利于工业化生产。
USPTO Abstract
本发明公开了用于制备4‑(2‐(4‐甲基苯基硫基))苯基哌啶的化合物、其制备方法及应用。本发明提供了两种制备4‑(2‐(4‐甲基苯基巯基))苯基哌啶的中间体:3‑(2‐(4‐甲基苯基巯基))苯基戊二酸和4‑(2‐(4‐甲基苯基巯基))苯基哌啶‐2,6‐二酮及其制备与应用。该方法收率高,操作安全、方便,对环境污染小且利于工业化生产。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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