CN Patent
CN104529904B — 玻玛西尼的制备方法
Assigned to Linyi High Tech Zone Jinlanling Labor Service Co ltd · Expires 2016-08-31 · 10y expired
What this patent protects
本发明揭示了一种玻玛西尼(Bemaciclib,亦称Abemaciclib)中间体及其制备方法,其制备步骤包括缩合、脒化及其环合等单元反应;以该玻玛西尼中间体为原料,经过胍基化反应和环合反应制得玻玛西尼。该制备方法原料易得,工艺简洁,经济环保,适合工业化生产。
USPTO Abstract
本发明揭示了一种玻玛西尼(Bemaciclib,亦称Abemaciclib)中间体及其制备方法,其制备步骤包括缩合、脒化及其环合等单元反应;以该玻玛西尼中间体为原料,经过胍基化反应和环合反应制得玻玛西尼。该制备方法原料易得,工艺简洁,经济环保,适合工业化生产。
Drugs covered by this patent
- Verzenio (abemaciclib) · Eli Lilly
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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