CN104163794A — 2-氨基芳环类血管内皮生长因子受体(vegfr)抑制剂及其制备方法和用途
Assigned to China Pharmaceutical University · Expires 2014-11-26 · 11y expired
What this patent protects
本发明涉及一种结构新颖的如式(I)所示的2-氨基吡啶类化合物、其药用盐、其前药、其水合物或溶剂合物,也涉及所述化合物的制备方法、包含治疗有效剂量的所述化合物的药物组合物,以及其作为蛋白酪氨酸激酶抑制剂,尤其是作为血管内皮生长因子-2-Vascular Endothelial Growth Factor Receptor2,VEGFR-2,Kinase Domain Receptor,KDR)抑制剂,在制备预防和/或治疗VEGFR-2异常相关疾病的药物中的用途。
USPTO Abstract
本发明涉及一种结构新颖的如式(I)所示的2-氨基吡啶类化合物、其药用盐、其前药、其水合物或溶剂合物,也涉及所述化合物的制备方法、包含治疗有效剂量的所述化合物的药物组合物,以及其作为蛋白酪氨酸激酶抑制剂,尤其是作为血管内皮生长因子-2-Vascular Endothelial Growth Factor Receptor2,VEGFR-2,Kinase Domain Receptor,KDR)抑制剂,在制备预防和/或治疗VEGFR-2异常相关疾病的药物中的用途。
Drugs covered by this patent
- Balversa (ERDAFITINIB) · Johnson & Johnson
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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