CN103910719B — 葡萄糖衍生物与苯丙氨酸复合物、晶体、制备方法及应用
Assigned to Shanghua Kechuang Investment Management Jiangsu Co ltd · Expires 2018-05-01 · 8y expired
What this patent protects
本发明公开了葡萄糖衍生物与苯丙氨酸复合物、晶体、制备方法及应用。化合物A·L‑苯丙氨酸复合物的共晶晶体的X‑射线粉末衍射,当衍射角为2θ时,在11.233,11.72,14.514,16.805,17.389,18.062,18.781,19.942,20.75,21.841,22.455,23.627,24.04,24.937,28.083,29.752和33.668处有特征峰。上述共晶晶体在制备治疗和/或预防由钠依赖的葡萄糖转运蛋白SGLT引起的疾病和/或症状、治疗和/或预防代谢失调症、治疗和/或预防胰腺β‑细胞的退化,或用于改善和/或恢复胰腺β‑细…
USPTO Abstract
本发明公开了葡萄糖衍生物与苯丙氨酸复合物、晶体、制备方法及应用。化合物A·L‑苯丙氨酸复合物的共晶晶体的X‑射线粉末衍射,当衍射角为2θ时,在11.233,11.72,14.514,16.805,17.389,18.062,18.781,19.942,20.75,21.841,22.455,23.627,24.04,24.937,28.083,29.752和33.668处有特征峰。上述共晶晶体在制备治疗和/或预防由钠依赖的葡萄糖转运蛋白SGLT引起的疾病和/或症状、治疗和/或预防代谢失调症、治疗和/或预防胰腺β‑细胞的退化,或用于改善和/或恢复胰腺β‑细胞功能性疾病的药物中的应用。
Drugs covered by this patent
- Farxiga (DAPAGLIFLOZIN) · AstraZeneca
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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