CN103804323A — 一种卡巴他赛溶剂化物及其制备方法和应用
Assigned to Aopudun (shanghai) Medical Technology Co Ltd · Expires 2014-05-21 · 12y expired
What this patent protects
本发明公开了一种卡巴他赛溶剂化物及其制备方法和应用。所述溶剂化物是由卡巴他赛与乙酸乙酯发生溶剂化后形成的结晶体,含有质量比为8~10%的乙酸乙酯。本发明提供的卡巴他赛溶剂化物具有稳定性好且吸湿性弱等优点,有利于制备质量符合标准的制剂;且其制备方法具有操作简单、质量稳定、得率高、成本低、节能环保等显著优点,符合工业化生产要求,具有极强的实用价值和广阔的应用前景。
USPTO Abstract
本发明公开了一种卡巴他赛溶剂化物及其制备方法和应用。所述溶剂化物是由卡巴他赛与乙酸乙酯发生溶剂化后形成的结晶体,含有质量比为8~10%的乙酸乙酯。本发明提供的卡巴他赛溶剂化物具有稳定性好且吸湿性弱等优点,有利于制备质量符合标准的制剂;且其制备方法具有操作简单、质量稳定、得率高、成本低、节能环保等显著优点,符合工业化生产要求,具有极强的实用价值和广阔的应用前景。
Drugs covered by this patent
- Jevtana Kit (cabazitaxel) · Accord Hlthcare
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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