CN Patent
CN103772449B — C‑芳基葡萄糖苷衍生物及其制备方法与用途
Assigned to Chang'ao Pharmaceutical Technology Holdings Ltd · Expires 2017-12-26 · 8y expired
What this patent protects
本发明公开了一种通式(I)所示的C‑芳基葡萄糖苷衍生物,其制备方法及用途,其中,R 1 、R 2 如说明书中所定义。所述的C‑芳基葡萄糖苷衍生物结构新颖,对SGLT‑2具有很强的抑制活性,同时对SGLT‑1和SGLT‑2的选择比也较高,可用于制备治疗和预防与钠依赖性葡萄糖转运蛋白相关疾病的药物。
USPTO Abstract
本发明公开了一种通式(I)所示的C‑芳基葡萄糖苷衍生物,其制备方法及用途,其中,R 1 、R 2 如说明书中所定义。所述的C‑芳基葡萄糖苷衍生物结构新颖,对SGLT‑2具有很强的抑制活性,同时对SGLT‑1和SGLT‑2的选择比也较高,可用于制备治疗和预防与钠依赖性葡萄糖转运蛋白相关疾病的药物。
Drugs covered by this patent
- Steglatro (ERTUGLIFLOZIN) · Merck & Co.
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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