CN Patent
CN103079544A — 包含丁丙诺啡的可注射的可流动组合物
Assigned to Rb Pharmaceutical Co ltd · Expires 2013-05-01 · 13y expired
What this patent protects
本发明涉及一种能够持续约14天至约3个月递送丁丙诺啡、其代谢产物或其前药的丁丙诺啡缓释递送体系。所述丁丙诺啡缓释递送体系包含用于缓释丁丙诺啡、其代谢产物或其前药的可流动组合物和固体植入物。所述植入物从所述可流动物组合物制得。所述丁丙诺啡缓释递送体系原位提供1个月和3个月的释放曲线,其特征在于极高的生物利用度和最低的永久性组织损伤风险,而且通常没有肌肉坏死的风险。
USPTO Abstract
本发明涉及一种能够持续约14天至约3个月递送丁丙诺啡、其代谢产物或其前药的丁丙诺啡缓释递送体系。所述丁丙诺啡缓释递送体系包含用于缓释丁丙诺啡、其代谢产物或其前药的可流动组合物和固体植入物。所述植入物从所述可流动物组合物制得。所述丁丙诺啡缓释递送体系原位提供1个月和3个月的释放曲线,其特征在于极高的生物利用度和最低的永久性组织损伤风险,而且通常没有肌肉坏死的风险。
Drugs covered by this patent
- Subutex (BUPRENORPHINE) · Purdue Pharma Lp
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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