CN Patent

CN102911169B — 一种卢拉西酮的制备方法

Assigned to Shanghai Institute of Pharmaceutical Industry · Expires 2015-05-06 · 11y expired

What this patent protects

本发明公开了一种如式I所示的卢拉西酮的制备方法,其包括下列步骤:在极性非质子溶剂中,在碱的作用下,将化合物II或化合物III,与化合物IV在50~150℃下进行如下反应,即可;本发明的卢拉西酮的制备方法收率高、操作简便、成本低,适合于工业上大规模生产,为卢拉西酮的制备提供了一条新的途径。

USPTO Abstract

本发明公开了一种如式I所示的卢拉西酮的制备方法,其包括下列步骤:在极性非质子溶剂中,在碱的作用下,将化合物II或化合物III,与化合物IV在50~150℃下进行如下反应,即可;本发明的卢拉西酮的制备方法收率高、操作简便、成本低,适合于工业上大规模生产,为卢拉西酮的制备提供了一条新的途径。

Drugs covered by this patent

Patent Metadata

Patent number
CN102911169B
Jurisdiction
CN
Classification
Expires
2015-05-06
Drug substance claim
No
Drug product claim
No
Assignee
Shanghai Institute of Pharmaceutical Industry
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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