CN102885792A — 盐酸西那卡塞的口服固体速释制剂
Assigned to China Resources Saike Pharmaceutical Co Ltd · Expires 2013-01-23 · 13y expired
What this patent protects
本发明公开了一种盐酸西那卡塞的口服固体速释制剂,包括盐酸西那卡塞和药用辅料,盐酸西那卡塞的平均粒径为5μm~15μm;所述盐酸西那卡塞为针状结晶性微粒;所述药用辅料包括填充剂、黏合剂、崩解剂和润滑剂;制剂形式为片剂。本发明有益效果:本发明通过对控制盐酸西那卡塞平均粒径的限定,提高了西那卡塞的溶出速率和溶出量,不仅制备工艺简单、安全,而且质量可控、成本低,适合工业化生产。
USPTO Abstract
本发明公开了一种盐酸西那卡塞的口服固体速释制剂,包括盐酸西那卡塞和药用辅料,盐酸西那卡塞的平均粒径为5μm~15μm;所述盐酸西那卡塞为针状结晶性微粒;所述药用辅料包括填充剂、黏合剂、崩解剂和润滑剂;制剂形式为片剂。本发明有益效果:本发明通过对控制盐酸西那卡塞平均粒径的限定,提高了西那卡塞的溶出速率和溶出量,不仅制备工艺简单、安全,而且质量可控、成本低,适合工业化生产。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
Track this patent
Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.