CN Patent

CN102885792A — 盐酸西那卡塞的口服固体速释制剂

Assigned to China Resources Saike Pharmaceutical Co Ltd · Expires 2013-01-23 · 13y expired

What this patent protects

本发明公开了一种盐酸西那卡塞的口服固体速释制剂,包括盐酸西那卡塞和药用辅料,盐酸西那卡塞的平均粒径为5μm~15μm;所述盐酸西那卡塞为针状结晶性微粒;所述药用辅料包括填充剂、黏合剂、崩解剂和润滑剂;制剂形式为片剂。本发明有益效果:本发明通过对控制盐酸西那卡塞平均粒径的限定,提高了西那卡塞的溶出速率和溶出量,不仅制备工艺简单、安全,而且质量可控、成本低,适合工业化生产。

USPTO Abstract

本发明公开了一种盐酸西那卡塞的口服固体速释制剂,包括盐酸西那卡塞和药用辅料,盐酸西那卡塞的平均粒径为5μm~15μm;所述盐酸西那卡塞为针状结晶性微粒;所述药用辅料包括填充剂、黏合剂、崩解剂和润滑剂;制剂形式为片剂。本发明有益效果:本发明通过对控制盐酸西那卡塞平均粒径的限定,提高了西那卡塞的溶出速率和溶出量,不仅制备工艺简单、安全,而且质量可控、成本低,适合工业化生产。

Drugs covered by this patent

Patent Metadata

Patent number
CN102885792A
Jurisdiction
CN
Classification
Expires
2013-01-23
Drug substance claim
No
Drug product claim
No
Assignee
China Resources Saike Pharmaceutical Co Ltd
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

Track this patent

Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.