CN Patent
CN102884066A — 8-氟-2-{4-[(甲氨基)甲基]苯基}-1,3,4,5-四氢-6H-氮杂*并[5,4,3-cd]吲哚-6-酮的盐和多晶型物
Assigned to Pfizer Inc · Expires 2013-01-16 · 13y expired
What this patent protects
本发明涉及8-氟-2-{4-[(甲氨基)甲基]苯基}-1,3,4,5-四氢-6H-氮杂 并[5,4,3-cd]吲哚-6-酮(式I)的新的多晶型形式及其制备方法。此类多晶型形式可以是药物组合物的成分,并且可用于治疗由聚(ADP-核糖)聚合酶活性所介导的哺乳动物疾病病状,包括诸如癌症的疾病病状。
USPTO Abstract
本发明涉及8-氟-2-{4-[(甲氨基)甲基]苯基}-1,3,4,5-四氢-6H-氮杂 并[5,4,3-cd]吲哚-6-酮(式I)的新的多晶型形式及其制备方法。此类多晶型形式可以是药物组合物的成分,并且可用于治疗由聚(ADP-核糖)聚合酶活性所介导的哺乳动物疾病病状,包括诸如癌症的疾病病状。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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