CN Patent
CN102186465B — 反胺苯环醇与nsaid的共晶
Assigned to Esteven Pharmaceutical Co ltd · Expires 2015-09-16 · 11y expired
What this patent protects
本发明涉及反胺苯环醇和选自NSAID的共晶前体的共晶、其制备方法及其作为药物或在药物制剂中的用途,尤其是用于治疗疼痛的用途。在一种优选实施方式中,该共晶是(-)-反胺苯环醇和(S)-萘普生(1∶2)的共晶;(+)-反胺苯环醇和(R)-萘普生(1∶2)的共晶或(外消旋)-盐酸反胺苯环醇-塞来昔布(1∶1)的共晶。
USPTO Abstract
本发明涉及反胺苯环醇和选自NSAID的共晶前体的共晶、其制备方法及其作为药物或在药物制剂中的用途,尤其是用于治疗疼痛的用途。在一种优选实施方式中,该共晶是(-)-反胺苯环醇和(S)-萘普生(1∶2)的共晶;(+)-反胺苯环醇和(R)-萘普生(1∶2)的共晶或(外消旋)-盐酸反胺苯环醇-塞来昔布(1∶1)的共晶。
Drugs covered by this patent
- Celebrex (celecoxib) · Pfizer Inc. (originally Searle/Pharmacia)
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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