CN Patent
CN102146059A — 喹唑啉衍生物、制备方法及其应用
Assigned to Shanghai Allist Pharmaceuticals Inc · Expires 2011-08-10 · 15y expired
What this patent protects
本发明公开了一种作为酪氨酸激酶不可逆抑制剂的喹唑啉衍生物,以及这类衍生物作为人类表皮生长因子受体(EGFR)突变体T790M的抑制剂和抗癌剂的应用。本发明还涉及其制备方法,以及一种包含喹唑啉衍生物的药物组合物。
USPTO Abstract
本发明公开了一种作为酪氨酸激酶不可逆抑制剂的喹唑啉衍生物,以及这类衍生物作为人类表皮生长因子受体(EGFR)突变体T790M的抑制剂和抗癌剂的应用。本发明还涉及其制备方法,以及一种包含喹唑啉衍生物的药物组合物。
Drugs covered by this patent
- Vizimpro (Dacomitinib) · Pfizer Inc.
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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