CN Patent

CN102093364B — 作为FAK/Pyk2抑制剂的2,4-二氨基-6,7-二氢-5H-吡咯并[2,3]嘧啶衍生物

Assigned to Centaurus Biopharma Co Ltd · Expires 2015-01-28 · 11y expired

What this patent protects

本发明公开了作为FAK/Pyk2抑制剂的由式(I)表示的2,4-二氨基-6,7-二氢-5H-吡咯并[2,3]嘧啶衍生物、或其药学上可接受的盐、溶剂化物、多晶型物、互变异构体或前药。本发明还公开了含有上述物质的药物组合物、其在制备药物中的应用以及用于治疗FAK和/或Pyk2介导的疾病或病症的方法。

USPTO Abstract

本发明公开了作为FAK/Pyk2抑制剂的由式(I)表示的2,4-二氨基-6,7-二氢-5H-吡咯并[2,3]嘧啶衍生物、或其药学上可接受的盐、溶剂化物、多晶型物、互变异构体或前药。本发明还公开了含有上述物质的药物组合物、其在制备药物中的应用以及用于治疗FAK和/或Pyk2介导的疾病或病症的方法。

Drugs covered by this patent

Patent Metadata

Patent number
CN102093364B
Jurisdiction
CN
Classification
Expires
2015-01-28
Drug substance claim
No
Drug product claim
No
Assignee
Centaurus Biopharma Co Ltd
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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