CN102078306A — 一种含有重组人血白蛋白的紫杉醇纳米颗粒冷冻干燥制剂
Assigned to WUXI YUANRONG BIOMEDICINE Co Ltd · Expires 2011-06-01 · 15y expired
What this patent protects
本发明公开一种含有重组人血白蛋白的纳米颗粒冷冻干燥粉末制剂,所述制剂由紫杉醇、磷脂、重组人血白蛋白、冻干支持剂和PH调节剂组成,各组分质量百分比如下:紫杉醇0.05-5%、磷脂0.1-50%、重组人血白蛋白1-60%、冻干支持剂1-60%、PH调节剂0.05-10%。本发明获得的纳米颗粒平均粒径小于0.4um,获得的粉末制剂和注射用水、葡萄糖和生理盐水重制形成PH在5.0-7.0之间的可注射水溶液,大大提高了该制剂的产业化价值。
USPTO Abstract
本发明公开一种含有重组人血白蛋白的纳米颗粒冷冻干燥粉末制剂,所述制剂由紫杉醇、磷脂、重组人血白蛋白、冻干支持剂和PH调节剂组成,各组分质量百分比如下:紫杉醇0.05-5%、磷脂0.1-50%、重组人血白蛋白1-60%、冻干支持剂1-60%、PH调节剂0.05-10%。本发明获得的纳米颗粒平均粒径小于0.4um,获得的粉末制剂和注射用水、葡萄糖和生理盐水重制形成PH在5.0-7.0之间的可注射水溶液,大大提高了该制剂的产业化价值。
Drugs covered by this patent
- Rapamune (sirolimus) · Pfizer
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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