CN102048734A — 药物组合物
Assigned to Sumitomo Pharma Co Ltd · Expires 2011-05-11 · 15y expired
What this patent protects
本发明涉及药物组合物。本发明涉及一种口服给药制剂,该制剂含有:预糊化淀粉,其含有通式(1)所示的N-[4-[4-(1,2-苯并异噻唑-3-基)-1-哌嗪基]-(2R,3R)-2,3-四亚甲基-丁基]-(1’R,2’S,3’R,4’S)-2,3-双环[2,2,1]庚烷二酰亚胺·盐酸盐(lurasidone)作为活性成分;水溶性赋型剂;水溶性聚合物粘合剂,所述制剂具有恒定的溶出特性,即使其活性成分的含量发生变化时也是如此。
USPTO Abstract
本发明涉及药物组合物。本发明涉及一种口服给药制剂,该制剂含有:预糊化淀粉,其含有通式(1)所示的N-[4-[4-(1,2-苯并异噻唑-3-基)-1-哌嗪基]-(2R,3R)-2,3-四亚甲基-丁基]-(1’R,2’S,3’R,4’S)-2,3-双环[2,2,1]庚烷二酰亚胺·盐酸盐(lurasidone)作为活性成分;水溶性赋型剂;水溶性聚合物粘合剂,所述制剂具有恒定的溶出特性,即使其活性成分的含量发生变化时也是如此。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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