CN Patent
CN101980704A — 选择性s1p1受体激动剂的给药方案
Assigned to Actelion Pharmaceuticals Ltd · Expires 2011-02-23 · 15y expired
What this patent protects
本发明涉及一种选择性S1P 1 受体激动剂的给药方案,其以下述方式将选择性S1P 1 受体激动剂施用至个体:在初始治疗期期间,以诱导心脏脱敏的剂量(该剂量低于目标剂量)及维持心脏脱敏的给药频率施用该选择性S1P 1 受体激动剂,直至不再发生急性心率降低,随后上调滴定剂量,至该选择性S1P 1 受体激动剂的目标剂量。
USPTO Abstract
本发明涉及一种选择性S1P 1 受体激动剂的给药方案,其以下述方式将选择性S1P 1 受体激动剂施用至个体:在初始治疗期期间,以诱导心脏脱敏的剂量(该剂量低于目标剂量)及维持心脏脱敏的给药频率施用该选择性S1P 1 受体激动剂,直至不再发生急性心率降低,随后上调滴定剂量,至该选择性S1P 1 受体激动剂的目标剂量。
Drugs covered by this patent
- Velsipity (Etrasimod Arginine) · Pfizer Inc.
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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