CN Patent
CN101653422A — 利培酮缓释微球、其制备方法和用途
Assigned to Nanjing Lvye Pharma Co Ltd · Expires 2010-02-24 · 16y expired
What this patent protects
本发明提供了一种利培酮缓释微球、其制备方法和用途。所述微球含有利培酮或9-羟基利培酮或其盐和未封端的丙交酯-乙交酯共聚物。本发明所提供的利培酮缓释微球具有更高的载药量,体内无突释现象、血药浓度平稳,且无药物释放停滞期,可以大大减少患者的给药频率,减少每次给药体积,提高了患者的顺应性,减少不良反应的发生。
USPTO Abstract
本发明提供了一种利培酮缓释微球、其制备方法和用途。所述微球含有利培酮或9-羟基利培酮或其盐和未封端的丙交酯-乙交酯共聚物。本发明所提供的利培酮缓释微球具有更高的载药量,体内无突释现象、血药浓度平稳,且无药物释放停滞期,可以大大减少患者的给药频率,减少每次给药体积,提高了患者的顺应性,减少不良反应的发生。
Drugs covered by this patent
- Risperdal (risperidone) · Johnson & Johnson (Janssen)
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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