CN Patent
CN101652139A — 药物组合物
Assigned to Daiichi Sankyo Co Ltd · Expires 2010-02-17 · 16y expired
What this patent protects
本发明提供在宽的pH范围内显示良好的溶出性的制剂。所述药物组合物含有:(A)下述式(1)表示的N 1 -(5-氯吡啶-2-基)-N 2 -((1S,2R,4S)-4-[(二甲基氨基)羰基]-2-{[(5-甲基-4,5,6,7-四氢噻唑并[5,4-c]吡啶-2-基)羰基]氨基)环己基)乙二酰胺、其药理上可接受的盐、或它们的水合物;和(B)选自糖醇类和水溶胀性添加剂中的1种或2种以上。
USPTO Abstract
本发明提供在宽的pH范围内显示良好的溶出性的制剂。所述药物组合物含有:(A)下述式(1)表示的N 1 -(5-氯吡啶-2-基)-N 2 -((1S,2R,4S)-4-[(二甲基氨基)羰基]-2-{[(5-甲基-4,5,6,7-四氢噻唑并[5,4-c]吡啶-2-基)羰基]氨基)环己基)乙二酰胺、其药理上可接受的盐、或它们的水合物;和(B)选自糖醇类和水溶胀性添加剂中的1种或2种以上。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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