CN Patent
CN101534818A — 用于治疗疼痛和脂类代谢疾病的氮杂环丁烷和氮杂环丁酮衍生物
Assigned to Merck Sharp and Dohme LLC · Expires 2009-09-16 · 17y expired
What this patent protects
本发明公开了式(I)化合物,其中Z 1 为-CH 2 -或-C(O)-,R 4 和R 5 为碳链(且任选可一起形成C 2 桥),u和v独立为0-3的整数,使得总和为3-5,R 2 为杂芳基,R 1 和R 3 如文中定义。本发明还公开了使用式(I)化合物治疗疼痛的方法。
USPTO Abstract
本发明公开了式(I)化合物,其中Z 1 为-CH 2 -或-C(O)-,R 4 和R 5 为碳链(且任选可一起形成C 2 桥),u和v独立为0-3的整数,使得总和为3-5,R 2 为杂芳基,R 1 和R 3 如文中定义。本发明还公开了使用式(I)化合物治疗疼痛的方法。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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