CN101268099A — 用于治疗性干预的y4选择性受体激动剂
Assigned to 7TM Pharma AS · Expires 2008-09-17 · 18y expired
What this patent protects
本说明书中所述的选自下组的Y4受体激动剂肽:[Ala30]PP 2-36 ,[Thr30]PP 2-36 ,Asn30]PP 2-36 ,[Gln30]PP 2-36 ,[Glu10]PP 2-36 ,[Glu10,Leu17,Thr30]PP 2-36 ,[Nle17,Nle30]PP 2-36 ,[Glu10,Nle17,Nle30]PP 2-36 ,它们的PP 1-36 等价物,以及它们的类似物和衍生物是相对于Y1和Y2受体的Y4受体选择性激动剂,可用于治疗肥胖症或超重,认为肥胖或超重是致病因素的疾病,以及腹泻和肠液分泌过多。
USPTO Abstract
本说明书中所述的选自下组的Y4受体激动剂肽:[Ala30]PP 2-36 ,[Thr30]PP 2-36 ,Asn30]PP 2-36 ,[Gln30]PP 2-36 ,[Glu10]PP 2-36 ,[Glu10,Leu17,Thr30]PP 2-36 ,[Nle17,Nle30]PP 2-36 ,[Glu10,Nle17,Nle30]PP 2-36 ,它们的PP 1-36 等价物,以及它们的类似物和衍生物是相对于Y1和Y2受体的Y4受体选择性激动剂,可用于治疗肥胖症或超重,认为肥胖或超重是致病因素的疾病,以及腹泻和肠液分泌过多。
Drugs covered by this patent
- Ozempic (semaglutide) · Novo Nordisk
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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